SCHEMBL21044489

SCHEMBL21044489

COC(=O)c1cc(CCCBr)cc(C(=O)OC)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
RECQL P46063 1/20 0.40
CYP4A11 Q02928 3/20 0.39
DAGLA Q9Y4D2 1/20 0.39
CYP4F2 P78329 2/20 0.38
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CES1 P23141 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.35
NQO2 P16083 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21044485 0.85 CYP4A11 (0.56) MAPTCYP1A2GAARECQLCYP4A11
SCHEMBL21044526 0.82 CYP4F2 (0.44) MAPTCYP1A2GAARECQLCYP4A11
SCHEMBL21044363 0.81 CYP4A11 (0.51) MAPTCYP1A2GAARECQLCYP4A11
SCHEMBL20886389 0.81 MAPK1 (0.41) MAPTCYP1A2GAARECQLMAPK1
SCHEMBL17595273 0.79 ALOX15 (0.47) MAPTCYP1A2KDM4EALDH1A1CES1
SCHEMBL20886358 0.78 GABRP (0.46) MAPTCYP1A2GAARECQLMAPK1
SCHEMBL17911801 0.77 MAPK1 (0.43) MAPTCYP1A2GAARECQLCYP4A11
SCHEMBL3597062 0.76 MAPK1 (0.53) MAPTCYP1A2CYP4A11CYP4F2MAPK1
SCHEMBL26162767 0.75 MTNR1A (0.38) MAPTCYP1A2GAARECQLMAPK1
SCHEMBL21044225 0.75 MAPK1 (0.42) MAPTCYP1A2GAARECQLMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191451-B1 4-SUBSTITUTED PYRIDINE-2,6-DICARBOXYLIC ACID DERIVATIVES AND METHOD OF PREPARING SAME OKINAWA INST SCIENCE & TECH SCHOOL CORP (JP) 2019-06-05 EP claimed