SCHEMBL21048820

SCHEMBL21048820

Cc1cnc(N(C)S(C)(=O)=O)c(CN(Cc2ccc([N+](=O)[O-])cc2)C(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.43
MMP1 P03956 2/20 0.41
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
MMP8 P22894 2/20 0.41
MMP13 P45452 2/20 0.41
CRHBP P24387 2/20 0.40
CRHR2 Q13324 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK4 Q16654 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21048818 0.79 MMP1 (0.42) MMP1MMP2MMP9MMP8MMP13
SCHEMBL17258964 0.72 CYP19A1 (0.44) CYP19A1CRHBPCRHR2CYP1A2CYP3A4
SCHEMBL17258961 0.72 CYP19A1 (0.44) CYP19A1CRHBPCRHR2CYP1A2CYP3A4
SCHEMBL11542075 0.72 CRHBP (0.68) MMP1MMP2MMP9MMP8MMP13
SCHEMBL21048923 0.70 PTK2 (0.49) ALDH1A1LMNASMN1; SMN2MEN1KMT2A
Acetic Acid SCHEMBL1627880 0.70 PTK2 (0.43) SMN1; SMN2
SCHEMBL12409792 0.68 PTK2 (0.43)
SCHEMBL1802673 0.67 CRHBP (0.60) CRHBPCRHR2CYP2C19ALDH1A1LMNA
Hydrochloric Acid SCHEMBL21048756 0.67 PTK2 (0.43)
SCHEMBL12640632 0.66 CRHBP (0.55) CYP19A1CRHBPCRHR2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed