SCHEMBL21048874

SCHEMBL21048874

CCN(c1ncc(F)cc1C#N)S(C)(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.35
SLC22A12 Q96S37 10/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
PTK2 Q05397 1/20 0.32
AR P10275 1/20 0.32
HDAC6 Q9UBN7 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17258959 0.83 ALDH1A1 (0.36) KDM4EALDH1A1TRPM8JAK2JAK1
SCHEMBL21048910 0.81 PTK2 (0.40) SLC22A12PTK2
Hydrochloric Acid SCHEMBL21048844 0.75 JAK2 (0.38) JAK2JAK1TYK2JAK3ALOX5AP
SCHEMBL1291285 0.74 PTK2 (0.40) KDM4EALDH1A1GAAHTTPTK2
SCHEMBL21048809 0.66 GAA (0.33) KDM4EALDH1A1SLC22A12CYP11B1CYP11B2
SCHEMBL1626886 0.65 PTK2 (0.37) KDM4EALDH1A1GAAHTTPTK2
SCHEMBL13082590 0.65 CHRNB2 (0.40) KDM4ESLC22A12CYP11B1CYP11B2JAK3
SCHEMBL17258736 0.64 PTK2 (0.36) KDM4EALDH1A1SLC22A12GAAHTT
SCHEMBL5495399 0.62 KDM4E (0.41) KDM4EALDH1A1SLC22A12CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL21048890 0.62 JAK2 (0.38) TRPM8JAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed