SCHEMBL21048880

SCHEMBL21048880

Cc1ccc(N(C)S(C)(=O)=O)c(CNC(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
PTK2 Q05397 2/20 0.46
JAK2 O60674 8/20 0.43
JAK1 P23458 8/20 0.43
TYK2 P29597 8/20 0.43
JAK3 P52333 8/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
NPSR1 Q6W5P4 1/20 0.40
HSPB1 P04792 1/20 0.40
CYP19A1 P11511 2/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17258747 0.86 ALDH1A1 (0.45) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL21048789 0.86 JAK2 (0.43) ALDH1A1PTK2JAK2JAK1TYK2
SCHEMBL21048852 0.83 ALDH1A1 (0.42) ALDH1A1PTK2JAK2JAK1TYK2
SCHEMBL21048855 0.83 JAK2 (0.44) ALDH1A1JAK2JAK1TYK2JAK3
SCHEMBL2181531 0.83 NPC1 (0.46) ALDH1A1NPC1RAB9AKMT2AGAA
SCHEMBL17258893 0.82 ALDH1A1 (0.53) ALDH1A1PTK2JAK2NPSR1KMT2A
SCHEMBL21048914 0.81 PTK2 (0.44) ALDH1A1PTK2JAK2JAK1TYK2
SCHEMBL16569947 0.80 ALDH1A1 (0.44) ALDH1A1PTK2JAK2JAK1TYK2
SCHEMBL21048876 0.79 PTK2 (0.43) ALDH1A1PTK2JAK2JAK1TYK2
SCHEMBL12409789 0.77 CYP19A1 (0.40) ALDH1A1PTK2JAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed