Lcl-161

Lcl-161

SCHEMBL21064744

CNC(C)C(=O)NC(C(=O)N1CCC[C@H]1c1nc(C(=O)c2ccc(F)cc2)cs1)C1CCCCC1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
XIAP P98170 15/20 0.50
RIPK2 O43353 12/20 0.50
ESR1 P03372 1/20 0.48
BIRC3 Q13489 3/20 0.46
BIRC2 Q13490 3/20 0.45
TRPV1 Q8NER1 1/20 0.42
TNF P01375 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lcl-161 SCHEMBL1275554 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
Lcl-161 SCHEMBL1275369 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
Lcl-161 SCHEMBL19164873 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
Lcl-161 SCHEMBL1275371 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
Lcl-161 SCHEMBL18663754 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
Lcl-161 SCHEMBL1495180 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
Lcl-161 SCHEMBL3688581 1.00 XIAP (0.50) XIAPRIPK2ESR1BIRC3BIRC2
SCHEMBL23975497 0.98 XIAP (0.49) XIAPRIPK2ESR1BIRC3BIRC2
SCHEMBL23975269 0.98 XIAP (0.49) XIAPRIPK2ESR1BIRC3BIRC2
SCHEMBL23975195 0.98 XIAP (0.49) XIAPRIPK2ESR1BIRC3BIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2296650-B1 IMMUNOMODULATION BY IAP INHIBITORS NOVARTIS AG (CH) 2020-05-06 EP claimed
US-10329626-B2 NOL3 is a predictor of patient outcome DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-06-25 US claimed
CN-101588801-B Combination of IAP inhibitors and FLT3 inhibitors NOVARTIS AG (CH) 2011-12-28 CN claimed
US-10975114-B2 Bis 2′-5′-RR-(3′F-A)(3′F-A) cyclic dinucleotide compound and uses thereof CHINOOK THERAPEUTICS, INC. (US) 2021-04-13 US disclosed
CN-111989338-A Modified cyclic dinucleotide compounds 勃林格殷格翰国际有限公司 2020-11-24 CN disclosed
US-20200199169-A1 BIS 2'-5'-RR-(3'F-A)(3'F-A) CYCLIC DINUCLEOTIDE COMPOUND AND USES THEREOF CHINOOK THERAPEUTICS, INC. 2020-06-25 US disclosed
EP-3116909-B1 ANTIBODY MOLECULES TO LAG-3 AND USES THEREOF NOVARTIS AG (CH) 2019-11-13 EP disclosed
CN-101588801-B Combination of IAP inhibitors and FLT3 inhibitors NOVARTIS AG (CH) 2011-12-28 CN disclosed
CN-101588801-A Combination of IAP inhibitors and FLT3 inhibitors NOVARTIS AG (CH) 2009-11-25 CN disclosed
CN-101541325-A Use of IAP inhibitors for the treatment of acute myeloid leukemia NOVARTIS AG (CH) 2009-09-23 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200199169-A1 BIS 2'-5'-RR-(3'F-A)(3'F-A) CYCLIC DINUCLEOTIDE COMPOUND AND USES THEREOF STING1, IRF3, IFNAR1 XIAP 1037/4885RIPK2 1070/4885ESR1 2028/4885
US-10329626-B2 NOL3 is a predictor of patient outcome MORF4L1, NOS3, NOS1 XIAP 1033/4885RIPK2 3353/4885ESR1 3116/4885
US-10975114-B2 Bis 2′-5′-RR-(3′F-A)(3′F-A) cyclic dinucleotide compound and uses thereof STING1, IRF3, IFNAR1 XIAP 1045/4885RIPK2 1061/4885ESR1 1971/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.