SCHEMBL21065872

SCHEMBL21065872

CC(=O)N1Cc2ccccc2/C=C(/C)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.54
HSD17B3 P37058 13/20 0.53
LMNA P02545 1/20 0.42
KCNN4 O15554 1/20 0.41
KCNA3 P22001 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26224571 0.89 HSD17B3 (0.44) NOTUMHSD17B3LMNAKCNN4KCNA3
SCHEMBL19889885 0.88 HSD17B3 (0.53) NOTUMHSD17B3
SCHEMBL19578541 0.86 KDM4E (0.56) NOTUMHSD17B3LMNAKCNN4KCNA3
SCHEMBL21604411 0.84 KDM4E (0.41) NOTUMHSD17B3LMNAKCNN4KCNA3
SCHEMBL24240781 0.80 NOTUM (0.55) NOTUMLMNA
SCHEMBL20202310 0.80 TSHR (0.39) NOTUMLMNA
SCHEMBL25009835 0.78 MTNR1A (0.42) LMNA
SCHEMBL27349417 0.78 DRD3 (0.38)
SCHEMBL25963738 0.78 NOTUM (0.60) NOTUMHSD17B3
SCHEMBL23659145 0.77 MAPT (0.39) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024146902-A1 METHODS OF PRODUCING HYDROGEL MICROSPHERES ASCENDIS PHARMA A/S (DK) 2024-07-11 WO disclosed
WO-2023141855-A1 PROTEIN CONJUGATES WITH MULTIPLE PAYLOADS AND METHODS FOR MAKING THE SAME GLYCO-THERAPY BIOTECHNOLOGY CO., LTD. (CN) 2023-08-03 WO disclosed
WO-2023141856-A1 CD3-TARGETING MULTISPECIFIC ANTIBODY AND USE THEREOF 岩唐生物科技(杭州)有限责任公司 2023-08-03 WO disclosed
WO-2023065137-A1 SITE-SPECIFIC GLYCOPROTEIN CONJUGATES AND METHODS FOR MAKING THE SAME GLYCO-THERAPY BIOTECHNOLOGY CO., LTD. (CN) 2023-04-27 WO disclosed
WO-2023011639-A1 OLIGOSACCHARIDE LINKER AND SIDE-CHAIN HYDROPHILIC FRAGMENT COMBINED GLYCOSITE-SPECIFIC ANTIBODY-DRUG CONJUGATE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海药物研究所 2023-02-09 WO disclosed
WO-2020112588-A1 ANTIBODY COMPRISING A GLUTAMINE-CONTAINING LIGHT CHAIN C-TERMINAL EXTENSION, CONJUGATES THEREOF, AND METHODS AND USES BRISTOL-MYERS SQUIBB COMPANY (US) 2020-06-04 WO disclosed
WO-2020028610-A1 2H-PYRAZOLO[4,3-d]PYRIMIDINE COMPOUNDS AS TOLL-LIKE RECEPTOR 7 (TLR7) AGONISTS AND METHODS AND USES THEREFOR BRISTOL-MYERS SQUIBB COMPANY (US) 2020-02-06 WO disclosed
EP-3134128-B1 SULFAMIDE LINKER, CONJUGATES THEREOF, AND METHODS OF PREPARATION SYNAFFIX BV (NL) 2019-06-05 EP disclosed