SCHEMBL210737

SCHEMBL210737

N#Cc1cccc(F)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT1 P54687 1/20 0.39
TSHR P16473 1/20 0.38
TRPV4 Q9HBA0 2/20 0.38
KHK P50053 1/20 0.37
AR P10275 5/20 0.37
DYRK1A Q13627 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
CUL4A Q13619 1/20 0.35
PDK2 Q15119 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30999675 1.00 BCAT1 (0.39) BCAT1TSHRTRPV4KHKAR
SCHEMBL3237062 0.83 TSHR (0.46) TSHRTRPV4ARDYRK1AESR2
SCHEMBL24084229 0.81 PDK2 (0.43) BCAT1ARESR2CA1CA2
SCHEMBL24084262 0.81 BCAT1 (0.43) BCAT1KHKESR2CA1CA2
SCHEMBL1365376 0.79 AR (0.46) TRPV4KHKARESR1ESR2
SCHEMBL2045858 0.77 CES2 (0.34) ARALDH1A1GAAALOX15
SCHEMBL16959428 0.77 TAAR1 (0.32) GAA
SCHEMBL101977 0.76 DYRK1A (0.47) TSHRTRPV4DYRK1ACA1CA2
SCHEMBL158537 0.76 BCAT1 (0.49) BCAT1TSHRTRPV4CA1CA2
SCHEMBL30443847 0.76 BCAT1 (0.49) BCAT1TSHRTRPV4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 116 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106883147-B A kind of preparation method of phenyl-pentafluoride formonitrile HCN 浙江工业大学 2018-11-02 CN claimed
CN-106883147-A A kind of preparation method of phenyl-pentafluoride formonitrile HCN 浙江工业大学 2017-06-23 CN claimed
CN-102603571-A Preparation method of 2,4-dichloro-3-cyano-5-fluobenzoic acid UNIV ZHEJIANG TECHNOLOGY 2012-07-25 CN claimed
CN-102531961-A Preparation method of 2,6-dichloro-3-fluorobenzonitrile UNIV ZHEJIANG TECHNOLOGY 2012-07-04 CN claimed
EP-0073372-B1 PROCESS FOR PRODUCING 2,6-DIFLUOROBENZONITRILE ISHIHARA SANGYO KAISHA, LTD. (JP) 1984-08-01 EP claimed
JP-1294653-A None JP disclosed
JP-1311052-A None JP disclosed
EP-4263544-B1 INDOLO[3.2.1-JK]CARBAZOLE-6-CARBONITRILE DERIVATIVES AS BLUE EMITTERS IN OLEDS UDC IRELAND LTD (IE) 2026-05-13 EP disclosed
US-20250243183-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS INCYTE CORPORATION 2025-07-31 US disclosed
US-12312331-B2 Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors INCYTE CORPORATION (US) 2025-05-27 US disclosed
US-20250100981-A1 Cis-substituted 5-(hydroxymethyl)morpholine-2-carboxamides as agonists of SSTR4 BOEHRINGER INGELHEIM INT (DE) 2025-03-27 US disclosed
WO-2025027049-A1 (2S,5R)-5-(HYDROXYMETHYL)MORPHOLINE-2-CARBOXAMIDES AS AGONISTS OF SSTR4 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-02-06 WO disclosed
EP-0270964-B1 PROCESS FOR OBTAINING SUBSTITUTED FLUOROBENZENES BAYER AG (DE) 1992-07-08 EP disclosed
EP-0372621-A1 Preparation of difluorobenzenes containing electron withdrawing substituents DowElanco (US) 1990-06-13 EP disclosed
JP-H01311052-A OPTICALLY ACTIVE COMPOUND AND USE THEREOF NIPPON TELEGR & TELEPH CORP <NTT> 1989-12-15 JP disclosed
JP-H01294653-A OPTICALLY ACTIVE LIQUID CRYSTAL COMPOUND NIPPON TELEGR & TELEPH CORP <NTT> 1989-11-28 JP disclosed
US-4868347-A SOLVENT EXTRACTION BAYER AKTIENGESELLSCHAFT (DE) 1989-09-19 US disclosed
EP-0270964-A2 Process for obtaining substituted fluorobenzenes BAYER AG (DE) 1988-06-15 EP disclosed
EP-0073372-B1 PROCESS FOR PRODUCING 2,6-DIFLUOROBENZONITRILE ISHIHARA SANGYO KAISHA, LTD. (JP) 1984-08-01 EP disclosed
US-4209457-A Production of halogenated benzonitriles I.S. C. Chemicals Limited (GB) 1980-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12312331-B2 Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors CDK2, CDK4, CDK2AP2 BCAT1 1254/4885TSHR 3599/4885TRPV4 4091/4885
US-20250100981-A1 Cis-substituted 5-(hydroxymethyl)morpholine-2-carboxamides as agonists of SSTR4 SSTR4, SSTR5, SSTR2 BCAT1 3580/4885TSHR 38/4885TRPV4 250/4885
US-20250243183-A1 IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS CDK2, CDK4, CDK2AP2 BCAT1 1254/4885TSHR 3599/4885TRPV4 4091/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.