SCHEMBL21076210

SCHEMBL21076210

C=CCc1ccc(N)c(-c2cc(CC=C)ccc2O)c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 13/20 0.79
GABRB2 P47870 13/20 0.79
CNR2 P34972 5/20 0.79
CNR1 P21554 4/20 0.79
MEN1 O00255 2/20 0.79
GAA P10253 2/20 0.79
MAPT P10636 2/20 0.79
KMT2A Q03164 2/20 0.79
ALDH1A1 P00352 2/20 0.79
KDM4E B2RXH2 1/20 0.79
ALDH2 P05091 1/20 0.79
AKR1B1 P15121 1/20 0.79
HPGD P15428 1/20 0.79
PPARG P37231 1/20 0.79
PPARD Q03181 1/20 0.79
NPSR1 Q6W5P4 1/20 0.79
TNKS O95271 1/20 0.66
PARP1 P09874 1/20 0.66
XDH P47989 1/20 0.59
ALOX5 P09917 6/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Magnolol SCHEMBL29538482 0.89 GABRA1 (1.00) GABRA1GABRB2CNR2CNR1MEN1
Magnolol SCHEMBL132477 0.89 GABRA1 (1.00) GABRA1GABRB2CNR2CNR1MEN1
SCHEMBL13577022 0.89 GABRA1 (0.59) GABRA1GABRB2CNR2CNR1MEN1
Magnolol SCHEMBL29649179 0.89 GABRA1 (1.00) GABRA1GABRB2CNR2CNR1MEN1
Randaiol SCHEMBL24922822 0.82 GABRA1 (0.85) GABRA1GABRB2CNR2CNR1MEN1
Magnolol SCHEMBL23119980 0.82 GABRA1 (0.85) GABRA1GABRB2CNR2CNR1MEN1
Randaiol SCHEMBL30114878 0.82 GABRA1 (0.85) GABRA1GABRB2CNR2CNR1MEN1
SCHEMBL30262895 0.82 TNKS (0.87) GABRA1GABRB2CNR2CNR1MEN1
SCHEMBL5139554 0.82 XDH (0.68) GABRA1GABRB2CNR2CNR1MEN1
SCHEMBL7762572 0.82 XDH (0.68) GABRA1GABRB2CNR2CNR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2753599-B1 BIPHENYL COMPOUNDS FOR USE IN TREATING MALARIA AND OTHER PARASITIC DISORDERS MEDIZINISCHE HOCHSCHULE HANNOVER (DE) 2019-06-05 EP disclosed