SCHEMBL21077862

SCHEMBL21077862

CCCN(CCC)C(=O)c1ccc(CC)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.62
EGFR P00533 2/20 0.58
ERBB2 P04626 2/20 0.58
HDAC1 Q13547 2/20 0.55
HDAC6 Q9UBN7 2/20 0.55
ALDH1A1 P00352 1/20 0.53
TP53 P04637 1/20 0.53
HPGD P15428 3/20 0.51
GABRA1 P14867 1/20 0.50
GABRB2 P47870 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
PLK1 P53350 1/20 0.48
POLB P06746 1/20 0.46
APEX1 P27695 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LPAR1 Q92633 1/20 0.46
LPAR5 Q9H1C0 1/20 0.46
LIMK1 P53667 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12309807 0.93 MLYCD (0.54) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL9694832 0.90 MLYCD (0.72) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL11919822 0.89 ALDH1A1 (0.50) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL10076244 0.87 ALDH1A1 (0.52) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL3559829 0.84 HPGD (0.61) MLYCDHDAC1HDAC6ALDH1A1HPGD
SCHEMBL12309792 0.83 ACACB (0.52) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL26314066 0.82 MLYCD (0.64) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL26313600 0.82 MLYCD (0.64) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL4489409 0.82 MLYCD (0.64) MLYCDEGFRERBB2HDAC1HDAC6
SCHEMBL7967022 0.82 MLYCD (0.64) MLYCDEGFRERBB2HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3694840-B1 PIPERAZINE DERIVATIVES AS MAGL INHIBITORS HOFFMANN LA ROCHE (CH) 2021-08-04 EP disclosed
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed