SCHEMBL10076244

SCHEMBL10076244

CCc1ccc(C(=O)N(CCO)CCO)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
HPGD P15428 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MLYCD O95822 2/20 0.47
PLK1 P53350 1/20 0.47
EGFR P00533 2/20 0.45
ERBB2 P04626 2/20 0.45
MAPT P10636 3/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
RAB9A P51151 1/20 0.43
LIMK2 P53671 1/20 0.43
THRA P10827 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12431478 0.93 HPGD (0.49) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1
SCHEMBL21077862 0.87 MLYCD (0.62) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1
SCHEMBL7157289 0.86 ALDH1A1 (0.48) ALDH1A1HPGDMLYCDEGFRERBB2
SCHEMBL11919822 0.84 ALDH1A1 (0.50) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1
SCHEMBL10076226 0.84 ALDH1A1 (0.50) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1
SCHEMBL3559829 0.82 HPGD (0.61) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1
SCHEMBL22851740 0.82 HPGD (0.44) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1
SCHEMBL19634427 0.81 HDAC3 (0.48) ALDH1A1MLYCDEGFRERBB2HDAC1
SCHEMBL7456186 0.81 ALDH1A1 (0.46) ALDH1A1HPGDSMN1; SMN2MLYCDEGFR
SCHEMBL12194867 0.81 MLYCD (0.58) ALDH1A1HPGDSMN1; SMN2MLYCDPLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093231-B2 Sulfonylethyl phosphorodiamidates TELIK, INC. (US) 2012-01-10 US disclosed
US-7879863-B2 Kallikrein inhibitors such as N-((2R)-3-methyl-2-{[4-(trifluoromethyl)phenyl]amino}butyl)-2-phenylacetamide trifluoroacetate, used for the treatment of gastrointestinal disorders, periodontal diseases, skin disorders, arthritis, hypotension, edema, respiratory system disorders and proliferative diseases AJINOMOTO CO., INC. (JP) 2011-02-01 US disclosed
US-20080039429-A1 SULFONYLETHYL PHOSPHORODIAMIDATES TELIK, INC. 2008-02-14 US disclosed
US-7262182-B2 Sulfonylethyl phosphorodiamidates TELIK, INC. (US) 2007-08-28 US disclosed
US-20070066586-A1 ANILINE DERIVATIVES AJINOMOTO CO., INC. (JP) 2007-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070066586-A1 ANILINE DERIVATIVES SERPINB1, ACE, REN ALDH1A1 747/4885HPGD 735/4885SMN1; SMN2 4457/4885
US-20080039429-A1 SULFONYLETHYL PHOSPHORODIAMIDATES MTAP, TYMP, PHOSPHO1 ALDH1A1 4455/4885HPGD 4123/4885SMN1; SMN2 1097/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.