SCHEMBL21078110

SCHEMBL21078110

N#CC1CCC(C(=O)N2CC=C(I)CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.37
JAK2 O60674 2/20 0.37
TYK2 P29597 1/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 1/20 0.34
NAMPT P43490 6/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
GRM5 P41594 1/20 0.33
KEAP1 Q14145 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRNB3 Q05901 1/20 0.33
CHRNA6 Q15825 1/20 0.33
PAX8 Q06710 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21078112 0.88 HPGD (0.42) JAK1JAK2TYK2ALDH1A1HPGD
SCHEMBL17888278 0.83 JAK1 (0.38) JAK1JAK2TYK2ALDH1A1HPGD
SCHEMBL21078144 0.82 KEAP1 (0.44) ALDH1A1HPGDNAMPTTSHRGRM5
SCHEMBL21077918 0.82 ALDH1A1 (0.48) ALDH1A1NAMPTTSHRKEAP1
SCHEMBL17886570 0.81 JAK1 (0.37) JAK1JAK2TYK2ALDH1A1HPGD
SCHEMBL21077905 0.81 ALDH1A1 (0.52) ALDH1A1HPGDNAMPTTSHRKEAP1
SCHEMBL21077917 0.78 NAMPT (0.48) ALDH1A1HPGDNAMPTKDM4EGRM5
SCHEMBL21078128 0.73 NAMPT (0.50) NAMPTGRM5
SCHEMBL21077851 0.72 JAK1 (0.35) JAK1JAK2ALDH1A1NAMPTKDM4E
SCHEMBL21078140 0.70 GRM5 (0.43) JAK1JAK2ALDH1A1NAMPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed