SCHEMBL21078902

SCHEMBL21078902

Cc1cc(C(=O)O)cnc1OCC(C)(C)C(F)F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 5/20 0.39
SSTR4 P31391 8/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
GABRA5 P31644 1/20 0.36
HCAR2 Q8TDS4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2714015 0.88 ALDH1A1 (0.43) AAK1SSTR4L3MBTL1CYP2C9CYP2C19
SCHEMBL21078799 0.86 L3MBTL1 (0.42) AAK1SSTR4L3MBTL1CYP2C9CYP2C19
SCHEMBL15350265 0.86 L3MBTL1 (0.42) AAK1SSTR4L3MBTL1CYP2C9CYP2C19
SCHEMBL2715676 0.84 L3MBTL1 (0.54) SSTR4L3MBTL1CYP2C9CYP2C19HCAR2
SCHEMBL2714128 0.81 SCN9A (0.39) L3MBTL1CYP2C9CYP2C19GABRA5HCAR2
SCHEMBL21078750 0.80 L3MBTL1 (0.40) AAK1SSTR4L3MBTL1CYP2C9CYP2C19
SCHEMBL15350077 0.79 L3MBTL1 (0.41) L3MBTL1CYP2C9CYP2C19HCAR2KDM4E
SCHEMBL15358626 0.78 L3MBTL1 (0.39) AAK1SSTR4L3MBTL1CYP2C9CYP2C19
SCHEMBL2716486 0.77 MAPK1 (0.41) AAK1SSTR4CYP2C9CYP2C19KDM4E
SCHEMBL21078829 0.77 CYP2C9 (0.40) L3MBTL1CYP2C9CYP2C19GABRA5HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2841421-B1 AMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2019-06-05 EP disclosed