SCHEMBL210903

SCHEMBL210903

CC(CC([NH])=O)N(Cc1ccc(F)cc1Cl)[C@H](COC(=O)Nc1cc2cc(F)ccc2cn1)CC(C)(C)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 9/20 0.34
AAK1 Q2M2I8 2/20 0.32
MAPK1 P28482 1/20 0.31
ROCK2 O75116 1/20 0.31
NR2C2 P49116 1/20 0.31
MAP2K1 Q02750 1/20 0.31
HIPK4 Q8NE63 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
BMP2K Q9NSY1 1/20 0.31
GSK3B P49841 3/20 0.31
DYRK1A Q13627 3/20 0.31
HTR2A P28223 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ALOX15 P16050 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
WNT1 P04628 1/20 0.30
CLK2 P49760 1/20 0.30
CLK3 P49761 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL213284 0.94 ABL1 (0.34) ABL1AAK1MAPK1ROCK2NR2C2
SCHEMBL213219 0.86 ABL1 (0.33) ABL1MAPK1GSK3BDYRK1AALDH1A1
SCHEMBL210902 0.81 P2RX7 (0.36) ABL1
SCHEMBL212353 0.81 P2RX7 (0.36) ABL1ROCK2
SCHEMBL211683 0.81 ABL1 (0.33) ABL1MAPK1GSK3BDYRK1AALDH1A1
SCHEMBL213218 0.79 P2RX7 (0.37)
SCHEMBL2722222 0.78 ABL1 (0.38) ABL1
SCHEMBL209990 0.76 P2RX7 (0.37) ABL1ALDH1A1ALOX15NPSR1HSD17B10
SCHEMBL213283 0.75 NPC1 (0.35) ABL1MAPK1ALDH1A1
SCHEMBL211931 0.75 ANO1 (0.36) ABL1MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8759374-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2014-06-24 US claimed
US-20120135964-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS QIAN XIANGPING (US) 2012-05-31 US claimed
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120135964-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS MYLK, MYH2, MYH10 ABL1 956/4885AAK1 4260/4885MAPK1 2926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.