SCHEMBL21090979

SCHEMBL21090979

CCCc1cc(CC)nc(C)n1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 3/20 0.48
NOS3 P29474 2/20 0.48
NOS1 P29475 1/20 0.48
BACE1 P56817 1/20 0.40
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP1A2 P05177 1/20 0.37
CTSK P43235 5/20 0.36
KDM5B Q9UGL1 1/20 0.35
CTSS P25774 3/20 0.35
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PDE10A Q9Y233 1/20 0.33
SREBF2 Q12772 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10051193 0.88 NOS3 (0.50) NOS2NOS3NOS1MAPTKDM5B
SCHEMBL13026558 0.82 NOS2 (0.48) NOS2NOS3NOS1BACE1MAPT
SCHEMBL1187597 0.79 NOS2 (0.57) NOS2NOS3NOS1CYP1A2NPSR1
SCHEMBL3802657 0.78 ALDH1A1 (0.46) NOS2NOS3NOS1BACE1MAPT
SCHEMBL9310993 0.78 NOS2 (0.46) NOS2NOS3NOS1BACE1MAPT
SCHEMBL1187650 0.77 KCNH2 (0.52) NOS2NOS3NOS1ALDH1A1
SCHEMBL805465 0.76 NOS3 (0.45) NOS2NOS3NOS1MAPTHSD17B10
SCHEMBL1188625 0.76 KCNH2 (0.55) NOS2NOS3NOS1ALDH1A1
SCHEMBL1187318 0.76 KCNH2 (0.55) NOS2NOS3NOS1ALDH1A1
SCHEMBL1188792 0.76 KCNH2 (0.55) NOS2NOS3NOS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108409672-B Method for synthesizing polysubstituted pyrimidine under catalysis of copper salt 安徽师范大学 2020-01-10 CN disclosed
EP-3495358-A1 AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFN ALPHA RESPONSES Bristol-Myers Squibb Company (US) 2019-06-12 EP disclosed