SCHEMBL21092244

SCHEMBL21092244

COC(=O)COc1ccc(C2CCOc3ccccc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 1/20 0.45
GLA P06280 1/20 0.41
CYP1A2 P05177 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.40
PPARD Q03181 1/20 0.39
PTGS2 P35354 1/20 0.39
ALOX5AP P20292 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21092019 0.87 ALOX15 (0.46) ESR1ESR2MEN1KMT2AALDH1A1
SCHEMBL20856119 0.80 CYP19A1 (0.51) MEN1KMT2AALDH1A1KDM4EMAPT
SCHEMBL11750596 0.75 CYP1A2 (0.48) ALDH1A1HPGDCYP1A2KDM4E
SCHEMBL11749703 0.75 MAPK1 (0.63) MEN1KMT2AALDH1A1CYP1A2POLB
SCHEMBL6479522 0.74 PIK3CA (0.37)
SCHEMBL11752378 0.74 GABRA1 (0.34) ESR1ESR2CYP1A2MAPT
SCHEMBL11752698 0.74 MAPK1 (0.41) MEN1KMT2AKDM4EMAPT
SCHEMBL11726825 0.74 CYP19A1 (0.38) PPARD
SCHEMBL11754929 0.74 ABL1 (0.35) ESR1ESR2
SCHEMBL11752049 0.73 MAPK1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817299-B1 SUBSTITUTED CHROMAN COMPOUNDS AS CALCIUM SENSING RECEPTOR MODULATORS LUPIN LTD (IN) 2019-06-12 EP disclosed