SCHEMBL21092019

SCHEMBL21092019

O=C(O)COc1ccc([C@@H]2CCOc3ccccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.46
PTPN7 P35236 2/20 0.43
FFAR1 O14842 2/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
CYP1A2 P05177 1/20 0.43
PPARG P37231 4/20 0.43
PPARD Q03181 4/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
PTPN12 Q05209 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.41
PPARA Q07869 1/20 0.40
MPO P05164 1/20 0.40
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
BLM P54132 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21092244 0.87 ESR1 (0.46) MEN1KMT2ACYP1A2PPARDALDH1A1
SCHEMBL11726825 0.79 CYP19A1 (0.38) PPARGPPARD
SCHEMBL11750596 0.78 CYP1A2 (0.48) ALOX15CYP1A2PPARGALDH1A1PPARA
SCHEMBL11749703 0.78 MAPK1 (0.63) PTPN7MEN1KMT2ACYP1A2PPARG
SCHEMBL29543994 0.78 OPRD1 (0.43) MEN1KMT2AMAPTLMNA
SCHEMBL2485975 0.78 OPRD1 (0.43) MEN1KMT2AMAPTLMNA
SCHEMBL11746234 0.77 KDM4E (0.46) MEN1KMT2AALDH1A1POLB
SCHEMBL11752639 0.77 HTR1A (0.33)
SCHEMBL20856119 0.77 CYP19A1 (0.51) MEN1KMT2AALDH1A1MAPTNPC1
SCHEMBL11724770 0.76 LMNA (0.39) ALOX15ALDH1A1MAPTESR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817299-B1 SUBSTITUTED CHROMAN COMPOUNDS AS CALCIUM SENSING RECEPTOR MODULATORS LUPIN LTD (IN) 2019-06-12 EP disclosed