SCHEMBL21101104

SCHEMBL21101104

O=C(O)c1ccc(CN2CCC(CNC3CC3)CC2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.50
KDM1A O60341 3/20 0.47
DRD2 P14416 1/20 0.47
MAOB P27338 1/20 0.47
HTR2A P28223 1/20 0.47
SLC6A4 P31645 1/20 0.47
SCN5A Q14524 1/20 0.47
CXCR3 P49682 1/20 0.45
CHRM4 P08173 2/20 0.45
ALDH1A1 P00352 1/20 0.44
CCR3 P51677 2/20 0.43
ACHE P22303 1/20 0.43
CXCR4 P61073 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21101005 0.88 KDM1A (0.50) SIGMAR1KDM1ADRD2MAOBHTR2A
SCHEMBL12821564 0.83 KDM1A (0.73) KDM1ADRD2MAOBHTR2ASLC6A4
SCHEMBL12821566 0.83 KDM1A (0.73) KDM1ADRD2MAOBHTR2ASLC6A4
SCHEMBL12966211 0.83 SIGMAR1 (0.48) SIGMAR1DRD2CHRM4ALDH1A1CCR3
SCHEMBL19725557 0.81 KDM1A (0.67) KDM1ADRD2MAOBHTR2ASLC6A4
SCHEMBL21101194 0.80 MCHR1 (0.56) SIGMAR1KDM1ADRD2MAOBHTR2A
SCHEMBL21101342 0.80 CYP2D6 (0.60) SIGMAR1KDM1ADRD2MAOBHTR2A
SCHEMBL21101256 0.79 SIGMAR1 (0.52) SIGMAR1KDM1ADRD2MAOBHTR2A
SCHEMBL21101096 0.78 BCHE (0.62) SIGMAR1DRD2SLC6A4CXCR3ACHE
SCHEMBL21100977 0.77 ALDH1A1 (0.52) SIGMAR1KDM1ADRD2MAOBHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2688568-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2019-06-19 EP disclosed