SCHEMBL21100977

SCHEMBL21100977

O=C(O)c1ccccc1CN1CCC(CNC2CC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
CCR3 P51677 4/20 0.50
HRH1 P35367 1/20 0.50
KCNH2 Q12809 1/20 0.50
CXCR4 P61073 6/20 0.49
KDM1A O60341 3/20 0.47
DRD2 P14416 1/20 0.47
MAOB P27338 1/20 0.47
HTR2A P28223 1/20 0.47
SLC6A4 P31645 1/20 0.47
SCN5A Q14524 1/20 0.47
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.46
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
BACE1 P56817 1/20 0.44
SIGMAR1 Q99720 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12813733 0.83 KDM1A (0.70) KCNH2KDM1ADRD2MAOBHTR2A
SCHEMBL12813735 0.83 KDM1A (0.70) KCNH2KDM1ADRD2MAOBHTR2A
SCHEMBL14032714 0.81 ALDH1A1 (0.56) ALDH1A1CCR3HRH1KCNH2CXCR4
SCHEMBL21101178 0.79 ATM (0.62) ALDH1A1CXCR4POLBKMT2ASIGMAR1
SCHEMBL14032449 0.78 ACHE (0.60) ALDH1A1CCR3HRH1KCNH2DRD2
SCHEMBL28169202 0.78 CXCR4 (0.68) ALDH1A1CCR3CXCR4KDM1AMAOB
SCHEMBL21101342 0.78 CYP2D6 (0.60) CCR3HRH1KCNH2CXCR4KDM1A
SCHEMBL21101005 0.77 KDM1A (0.50) KCNH2CXCR4KDM1ADRD2MAOB
SCHEMBL21101104 0.77 SIGMAR1 (0.50) ALDH1A1CCR3CXCR4KDM1ADRD2
SCHEMBL19725557 0.76 KDM1A (0.67) CXCR4KDM1ADRD2MAOBHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2688568-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2019-06-19 EP disclosed