SCHEMBL21101616

SCHEMBL21101616

c1ccc(N2CCC(CNC3CC3)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.50
ADRA1A P35348 1/20 0.50
ADRA1B P35368 1/20 0.50
KDM1A O60341 4/20 0.49
TPSAB1 Q15661 1/20 0.47
MBTD1 Q05BQ5 1/20 0.46
L3MBTL3 Q96JM7 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
DRD2 P14416 5/20 0.45
DRD3 P35462 5/20 0.45
ACHE P22303 3/20 0.43
MAOB P27338 2/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
NPC1 O15118 1/20 0.43
CHRNA7 P36544 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10154050 0.81 ADRA1D (0.51) ADRA1DADRA1AADRA1BKDM1AMBTD1
SCHEMBL12813593 0.79 KDM1A (0.77) KDM1ADRD2MAOBSLC6A4
SCHEMBL12813596 0.79 KDM1A (0.77) KDM1ADRD2MAOBSLC6A4
SCHEMBL13798544 0.77 CHRNA7 (0.50) MBTD1L3MBTL3L3MBTL1DRD2ACHE
SCHEMBL4071616 0.77 ADRA1D (0.51) ADRA1DADRA1AADRA1BKDM1AMBTD1
SCHEMBL19700585 0.77 ADRA1D (0.48) ADRA1DADRA1AADRA1BKDM1AMBTD1
SCHEMBL28169202 0.77 CXCR4 (0.68) KDM1AACHEMAOB
SCHEMBL7841536 0.76 ACHE (0.66) ACHE
SCHEMBL24123852 0.75 ME3 (0.46) KDM1AMBTD1L3MBTL3L3MBTL1ACHE
SCHEMBL424881 0.74 CHRNA7 (0.55) MBTD1L3MBTL3L3MBTL1HRH3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2688568-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2019-06-19 EP disclosed