SCHEMBL21136934

SCHEMBL21136934

Cc1cc2c(O)c([N+](=O)[O-])cnc2cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
PKM P14618 2/20 0.41
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSP90AA1 P07900 1/20 0.41
OPRK1 P41145 1/20 0.41
GPR35 Q9HC97 4/20 0.40
PPIA P62937 1/20 0.36
PGK1 P00558 1/20 0.36
CYP3A4 P08684 1/20 0.36
CTSB P07858 1/20 0.35
GAA P10253 1/20 0.35
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21136767 0.85 PGK1 (0.38) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL21050923 0.83 MEN1 (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL16618826 0.83 CYP1A2 (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL21099305 0.80 MAPT (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL29970861 0.80 CYP1A2 (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL26131807 0.80 CYP1A2 (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL27846638 0.78 GPR35 (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL18249961 0.77 ERN1 (0.46) CYP3A4
SCHEMBL1025814 0.77 MAPT (0.48) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL5767153 0.77 GPR35 (0.46) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019110751-A1 TETRACYCLIC COMPOUNDS AS INHIBITORS OF G12C MUTANT RAS PROTEIN, FOR USE AS ANTI-CANCER AGENTS ASTRAZENECA AB (SE) 2019-06-13 WO disclosed