SCHEMBL21154673

SCHEMBL21154673

CC(C)Sc1ccc(F)cc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.40
KEAP1 Q14145 1/20 0.40
CES2 O00748 3/20 0.39
CES1 P23141 3/20 0.39
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
KCNE1 P15382 1/20 0.37
KCNQ1 P51787 1/20 0.37
PARP1 P09874 2/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
AGBL2 Q5U5Z8 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
JAK2 O60674 2/20 0.36
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
DGAT1 O75907 1/20 0.35
PARP14 Q460N5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20196932 0.81 KMT2A (0.41) CA2IRAK4ALDH1A1KMT2A
SCHEMBL9710337 0.80 KEAP1 (0.46) KEAP1CES2CES1PARP1JAK2
SCHEMBL6781811 0.75 SIRT1 (0.55) CA2KEAP1IRAK4NPC1RAB9A
SCHEMBL15082650 0.74 RECQL (0.44) KEAP1CES2CES1PARP1IRAK4
SCHEMBL29463969 0.72 CES2 (0.52) KEAP1CES2CES1PARP1JAK2
SCHEMBL10160070 0.71 POLB (0.45) KEAP1CES2CES1PARP1IRAK4
SCHEMBL2852106 0.71 KEAP1 (0.47) KEAP1CES2CES1PARP1NPC1
SCHEMBL4068010 0.70 CES2 (0.42) KEAP1CES2CES1PARP1RAB9A
SCHEMBL29537903 0.70 CES2 (0.68) KEAP1CES2CES1PARP1JAK2
SCHEMBL366058 0.70 CES2 (0.68) KEAP1CES2CES1PARP1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607950-A2 HEPATITIS B CORE PROTEIN ALLOSTERIC MODULATORS Indiana University Research & Technology Corporation (US) 2020-02-12 EP disclosed
EP-3116316-B1 HEPATITIS B CORE PROTEIN ALLOSTERIC MODULATORS UNIV INDIANA RES & TECH CORP (US) 2019-07-10 EP disclosed