SCHEMBL9710337

SCHEMBL9710337

NC(=O)c1cc(F)ccc1SSc1ccc(F)cc1C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
CES2 O00748 3/20 0.45
CES1 P23141 3/20 0.45
PARP1 P09874 2/20 0.42
DGAT1 O75907 1/20 0.40
IKBKB O14920 2/20 0.37
MEN1 O00255 1/20 0.37
JAK2 O60674 1/20 0.37
EIF2AK2 P19525 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
POLB P06746 1/20 0.36
MAPK8 P45983 2/20 0.36
LMNA P02545 1/20 0.36
CHUK O15111 1/20 0.36
CDC7 O00311 1/20 0.36
KCNN4 O15554 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9710267 0.84 CES2 (0.45) KEAP1CES2CES1PARP1DGAT1
SCHEMBL6227763 0.82 KEAP1 (0.57) KEAP1CES2CES1MEN1KMT2A
SCHEMBL21154673 0.80 CA2 (0.40) KEAP1CES2CES1PARP1DGAT1
SCHEMBL6225041 0.80 CES2 (0.45) KEAP1CES2CES1POLBALDH1A1
SCHEMBL29463969 0.79 CES2 (0.52) KEAP1CES2CES1PARP1DGAT1
SCHEMBL7017263 0.78 MAPT (0.47) IKBKBMEN1KMT2ATDP1POLB
SCHEMBL29537903 0.77 CES2 (0.68) KEAP1CES2CES1PARP1DGAT1
SCHEMBL366058 0.77 CES2 (0.68) KEAP1CES2CES1PARP1DGAT1
SCHEMBL11377040 0.76 KDM4E (0.53) PARP1ALDH1A1
SCHEMBL3916230 0.75 ALDH1A1 (0.50) KEAP1CES2CES1PARP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021668-A1 BENZOTHIAZEPINONES AND THEIR USE AS ANTICONVULSANTS THE BOOTS COMPANY PLC (GB) 1992-12-10 WO disclosed