SCHEMBL21154840

SCHEMBL21154840

CCOC(=O)c1cc(Br)c(CNCc2ccc(OC)cc2OC)cc1F

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.52
MAPT P10636 3/20 0.51
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 3/20 0.42
POLB P06746 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157655 0.80 MAPT (0.55) APLNRMAPTHTR2AHTR2CALDH1A1
SCHEMBL20912632 0.74 MAPT (0.55) APLNRMAPTALDH1A1POLBTDP1
SCHEMBL523291 0.74 APLNR (0.63) APLNRMAPTHTR2AHTR2CHDAC3
SCHEMBL21154838 0.73 CYP4F2 (0.44) MAPTKMT2AALDH1A1NPSR1TSHR
SCHEMBL23635828 0.73 HPGD (0.56) MAPTMEN1KMT2AALDH1A1RAB9A
SCHEMBL12093644 0.73 KDM4E (0.56) MAPTALDH1A1NPSR1RAB9ATSHR
SCHEMBL783785 0.72 APLNR (1.00) APLNRHTR2AHTR2CHDAC3HDAC1
SCHEMBL2225000 0.72 APLNR (0.60) APLNRMAPTHTR2AHTR2CHDAC3
SCHEMBL22852762 0.71 HPGD (0.57) MAPTMEN1KMT2AALDH1A1RAB9A
SCHEMBL7488349 0.71 KMT2A (0.67) HDAC3HDAC1HDAC2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019134680-A1 INHIBITOR OF APOPTOSIS SIGNAL-REGULATING KINASE-1 AND APPLICATION THEREOF 广州市恒诺康医药科技有限公司 2019-07-11 WO disclosed