SCHEMBL21155022

SCHEMBL21155022

CNC(=O)c1ccccc1Sc1ccc(C(=O)O)c(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.49
ALDH1A1 P00352 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
PLK1 P53350 1/20 0.47
NLRP3 Q96P20 1/20 0.46
SLC6A3 Q01959 3/20 0.45
SLC6A2 P23975 2/20 0.45
SLC6A4 P31645 2/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
KDR P35968 4/20 0.44
PLK4 O00444 2/20 0.44
AURKA O14965 2/20 0.44
MAP4K4 O95819 2/20 0.44
PAK4 O96013 2/20 0.44
ABL1 P00519 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18666776 0.83 SLC6A3 (0.48) ALDH1A1MEN1KMT2AL3MBTL1SLC6A3
SCHEMBL232284 0.81 HTT (0.50) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL6216437 0.78 NSD2 (0.44) HPGDALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8533409 0.78 CLCN2 (0.46) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL11750773 0.78 SIRT1 (0.61) HPGDALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL8612788 0.76 SLC6A3 (0.49) HPGDALDH1A1L3MBTL1PLK1SLC6A3
SCHEMBL18664358 0.75 RAB9A (0.56) HPGDALDH1A1KMT2AL3MBTL1SMN1; SMN2
SCHEMBL618503 0.73 SLC6A3 (0.54) HPGDKMT2AL3MBTL1PLK1SLC6A3
SCHEMBL22579323 0.72 SLC6A3 (0.45) PLK1SLC6A3SLC6A2SLC6A4KDR
SCHEMBL11442238 0.72 SIRT1 (0.46) HPGDALDH1A1KMT2AL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3116316-B1 HEPATITIS B CORE PROTEIN ALLOSTERIC MODULATORS UNIV INDIANA RES & TECH CORP (US) 2019-07-10 EP disclosed