SCHEMBL8533409

SCHEMBL8533409

COc1cc(Sc2ccccc2C(=O)O)ccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLCN2 P51788 2/20 0.46
PTPRG P23470 1/20 0.45
NSD2 O96028 1/20 0.44
ALDH1A1 P00352 4/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KCNH2 Q12809 1/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 2/20 0.43
AR P10275 1/20 0.43
POLB P06746 1/20 0.42
GRM4 Q14833 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CA12 O43570 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530235 0.89 AR (0.43) CLCN2ALDH1A1HTTNPC1RAB9A
SCHEMBL232284 0.87 HTT (0.50) NSD2ALDH1A1HTTNPC1RAB9A
SCHEMBL8533973 0.86 ALDH1A1 (0.60) ALDH1A1HTTNPC1RAB9AMEN1
SCHEMBL11478744 0.84 AKR1C3 (0.42) ALDH1A1NPC1MEN1KMT2AKDM4E
SCHEMBL6216437 0.84 NSD2 (0.44) NSD2ALDH1A1HTTNPC1RAB9A
SCHEMBL11472530 0.83 PTPRG (0.58) PTPRGNSD2ALDH1A1NPC1RAB9A
SCHEMBL11480340 0.81 MMP2 (0.60) HPGDARGRM4HDAC6ITGAL
SCHEMBL2707834 0.80 PRKAG1 (0.50) CLCN2PTPRGNSD2ALDH1A1HTT
SCHEMBL11473506 0.79 PTPRG (0.48) PTPRGNSD2ALDH1A1HTTNPC1
Hydrochloric Acid SCHEMBL10670862 0.78 ALDH1A1 (0.53) CLCN2PTPRGALDH1A1HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed
US-4238611-A Polysubstituted derivatives of 10-piperazinodibenzo (b,f) thiepine SPOFA, UNITED PHARMACEUTICAL WORKS (CS) 1980-12-09 US disclosed