SCHEMBL21156580

SCHEMBL21156580

CCOC(=O)c1cc2cc(-c3ncc[nH]3)cn2c(C(C)=O)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EED O75530 1/20 0.38
RBBP4 Q09028 1/20 0.38
SUZ12 Q15022 1/20 0.38
EZH2 Q15910 1/20 0.38
AEBP2 Q6ZN18 1/20 0.38
BRD4 O60885 1/20 0.38
KDM4E B2RXH2 9/20 0.37
ALDH1A1 P00352 6/20 0.37
NUDT1 P36639 1/20 0.37
HPGD P15428 4/20 0.34
GAA P10253 5/20 0.34
NPC1 O15118 2/20 0.34
POLB P06746 1/20 0.34
BAZ2B Q9UIF8 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33
GLA P06280 3/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 1/20 0.33
SMPD3 Q9NY59 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21113222 0.88 BRD4 (0.40) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL19964897 0.81 CASP1 (0.45) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL21113398 0.80 BAZ2B (0.39) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21113367 0.79 JMJD6 (0.44) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21113193 0.79 ALDH1A1 (0.38) KDM4EALDH1A1HPGDGAANPC1
SCHEMBL21113401 0.79 LMNA (0.41) BRD4KDM4EALDH1A1HPGDGAA
SCHEMBL29985958 0.79 LMNA (0.41) BRD4KDM4EALDH1A1HPGDGAA
SCHEMBL21113246 0.79 BAZ2B (0.38) KDM4EALDH1A1HPGDGAANPC1
SCHEMBL21113282 0.79 BAZ2B (0.37) KDM4EALDH1A1HPGDGAANPC1
SCHEMBL21113224 0.78 ALDH1A1 (0.44) KDM4EALDH1A1HPGDGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10968215-B2 Pyrido five-element aromatic ring compound, preparation method therefor and use thereof SHANGHAI HAIHE PHARMACEUTICAL CO., LTD. (CN) 2021-04-06 US disclosed
US-20190211010-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF HAIHE BIOPHARMA CO. LTD. (CN) 2019-07-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10968215-B2 Pyrido five-element aromatic ring compound, preparation method therefor and use thereof EZH2, IKZF2, SUZ12 EED 41/4885RBBP4 288/4885SUZ12 3/4885
US-20190211010-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF EZH2, IKZF2, SUZ12 EED 41/4885RBBP4 288/4885SUZ12 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.