SCHEMBL21163196

SCHEMBL21163196

CC(C)(C)OC(=O)N1CCC[C@H]1c1cc(C2CCCCCCCCCC2)no1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
TSHR P16473 6/20 0.41
USP30 Q70CQ3 3/20 0.41
LMNA P02545 4/20 0.41
NPSR1 Q6W5P4 3/20 0.41
MAPT P10636 2/20 0.41
HTT P42858 1/20 0.40
EPHX2 P34913 1/20 0.39
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21163197 0.91 ALDH1A1 (0.44) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL8114296 0.83 CHRNB2 (0.56) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL8121446 0.83 CHRNB2 (0.56) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL9254476 0.82 CHRNB2 (0.51) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL9264718 0.82 SCD5 (0.49) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL9264284 0.81 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL8121245 0.81 ALDH1A1 (0.48) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL8139425 0.81 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AL3MBTL1TSHR
SCHEMBL21163195 0.81 GRM5 (0.47)
SCHEMBL21065088 0.81 HCRTR1 (0.57) ALDH1A1TSHRUSP30LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906553-B1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO)ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2019-06-26 EP disclosed