SCHEMBL21170229

SCHEMBL21170229

C=C(N)c1cccc(-c2ccc(NCC(C)(C)c3ccccc3Cl)nn2)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IL1B P01584 5/20 0.37
NLRP3 Q96P20 1/20 0.36
KDM4A O75164 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
NPC1 O15118 1/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PHF8 Q9UPP1 1/20 0.33
ACHE P22303 3/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12289883 0.90 KDM4A (0.39) IL1BNLRP3KDM4AKDM5AKDM4C
SCHEMBL21170210 0.88 NPC1 (0.36) IL1BNLRP3NPC1USP2TP53
SCHEMBL21170233 0.84 IL1B (0.37) IL1BNLRP3NPC1USP2TP53
SCHEMBL21170422 0.83 IL1B (0.35) IL1BNLRP3NPC1USP2TP53
SCHEMBL12289888 0.81 CYP11B1 (0.38) IL1BNLRP3KDM4AKDM5AKDM4C
SCHEMBL21170296 0.81 IL1B (0.36) IL1BNLRP3NPC1USP2TP53
SCHEMBL21170105 0.80 IL1B (0.36) IL1BNLRP3NPC1USP2TP53
SCHEMBL21170329 0.78 IL1B (0.34) IL1BNLRP3NPC1USP2TP53
SCHEMBL12286720 0.78 NPC1 (0.40) IL1BNPC1RAB9ASMN1; SMN2
SCHEMBL2562880 0.78 SMN1; SMN2 (0.40) IL1BNPC1USP2TP53RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed