SCHEMBL21170422

SCHEMBL21170422

C=C(N)c1cccc(-c2ccc(NCC(C)(C)c3ncccn3)nn2)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IL1B P01584 10/20 0.35
NPC1 O15118 1/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
WNT3A P56704 1/20 0.32
MAP4K4 O95819 1/20 0.32
TNF P01375 1/20 0.32
NLRP3 Q96P20 1/20 0.32
GPR39 O43194 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12288240 0.89 MAPK8 (0.40)
SCHEMBL21170329 0.88 IL1B (0.34) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170105 0.84 IL1B (0.36) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170233 0.84 IL1B (0.37) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170210 0.83 NPC1 (0.36) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170229 0.83 IL1B (0.37) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170125 0.82 IL1B (0.35) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170296 0.81 IL1B (0.36) IL1BNPC1USP2TP53RAB9A
SCHEMBL21170275 0.79 IL1B (0.34) IL1BTNF
SCHEMBL12286826 0.77 PDE4A (0.38) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed