SCHEMBL21170210

SCHEMBL21170210

C=C(N)c1cccc(-c2ccc(NCC(C)(C)c3ccccc3F)nn2)c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
IL1B P01584 9/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
TNF P01375 1/20 0.32
SOAT2 O75908 1/20 0.32
SOAT1 P35610 1/20 0.32
NLRP3 Q96P20 1/20 0.32
MEN1 O00255 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
KMT2A Q03164 1/20 0.31
RELA Q04206 1/20 0.31
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12286720 0.90 NPC1 (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL21170296 0.89 IL1B (0.36) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL21170229 0.88 IL1B (0.37) NPC1RAB9ASMN1; SMN2IL1BUSP2
SCHEMBL21170329 0.86 IL1B (0.34) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL21170422 0.83 IL1B (0.35) NPC1RAB9ASMN1; SMN2IL1BUSP2
SCHEMBL21170125 0.82 IL1B (0.35) NPC1RAB9ASMN1; SMN2IL1BUSP2
SCHEMBL21170105 0.80 IL1B (0.36) NPC1RAB9ASMN1; SMN2IL1BUSP2
SCHEMBL21170233 0.80 IL1B (0.37) NPC1RAB9ASMN1; SMN2IL1BUSP2
SCHEMBL12287812 0.80 HPGDS (0.40) NPC1RAB9AALDH1A1TP53SOAT2
SCHEMBL12289883 0.78 KDM4A (0.39) IL1BNLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed