SCHEMBL21177161

SCHEMBL21177161

CCCOC(=O)c1oc(Cc2cc(F)c3ncc(Cl)cc3c2)nc1C#N

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 4/20 0.42
MAP4K1 Q92918 1/20 0.33
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177639 0.85 KLKB1 (0.45) KLKB1MAP4K1ALDH1A1TSHRMAPK1
SCHEMBL21177781 0.81 KLKB1 (0.36) KLKB1MAP4K1ALDH1A1MAPK1NPSR1
SCHEMBL21177327 0.78 S1PR1 (0.37) KLKB1ALDH1A1
SCHEMBL21180345 0.77 KLKB1 (0.40) KLKB1MAP4K1ALDH1A1TSHRMAPK1
SCHEMBL21177539 0.77 KLKB1 (0.40) KLKB1MAP4K1ALDH1A1TSHRMAPK1
SCHEMBL19779896 0.76 KLKB1 (0.62) KLKB1MAP4K1ALDH1A1
SCHEMBL21177362 0.75 KLKB1 (0.38) KLKB1MAP4K1ALDH1A1TSHR
SCHEMBL21177142 0.73 KLKB1 (0.36) KLKB1MAP4K1ALDH1A1
SCHEMBL19780407 0.73 KLKB1 (0.42) KLKB1MAPK1NPSR1
SCHEMBL21177545 0.71 KLKB1 (0.34) KLKB1MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed