SCHEMBL21180476

SCHEMBL21180476

CC(C)(C)OC(=O)NCC(=O)c1ccc(F)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.43
CHRNG P07510 1/20 0.43
CHRNB1 P11230 1/20 0.43
CHRNB2 P17787 1/20 0.43
SLC6A2 P23975 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CHRND Q07001 1/20 0.43
DPP4 P27487 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
TRPA1 O75762 1/20 0.41
EGFR P00533 1/20 0.39
AURKB Q96GD4 1/20 0.39
KDM4A O75164 1/20 0.39
SERPINE1 P05121 1/20 0.38
CYP17A1 P05093 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12497673 0.88 EGFR (0.48) EGFRAURKBTAS1R3TAS1R1TAS1R2
SCHEMBL22305299 0.87 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2POLB
SCHEMBL5955544 0.84 PLOD2 (0.46) DPP4ALDH1A1PKMTSHRSMN1; SMN2
SCHEMBL8558279 0.81 CA12 (0.46) KDM4ASERPINE1POLB
SCHEMBL14830379 0.81 ALDH1A1 (0.52) ALDH1A1PKMTSHRSMN1; SMN2MEN1
SCHEMBL882755 0.80 HDAC1 (0.44) KDM4ACYP17A1ALDH1A1PKMTSHR
SCHEMBL26921163 0.80 HPGD (0.47) ALDH1A1TSHRPOLBIDO1
SCHEMBL19331732 0.79 MAPT (0.51) KDM4AALDH1A1PKMTSHRSMN1; SMN2
SCHEMBL2009324 0.79 NR1H4 (0.47) ALDH1A1PKMTSHRSMN1; SMN2POLB
SCHEMBL23017662 0.79 ERCC5 (0.49) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260124204-A1 METALLOENZYME INHIBITOR COMPOUNDS EIKONIZO THERAPEUTICS, INC. (US) 2026-05-07 US disclosed
US-12370194-B2 Metalloenzyme inhibitor compounds EIKONIZO THERAPEUTICS, INC. (US) 2025-07-29 US disclosed
US-20240307391-A1 METALLOENZYME INHIBITOR COMPOUNDS EIKONIZO THERAPEUTICS, INC. (US) 2024-09-19 US disclosed
US-11938134-B2 Metalloenzyme inhibitor compounds EIKONIZO THERAPEUTICS, INC. (US) 2024-03-26 US disclosed
US-20220088018-A1 METALLOENZYME INHIBITOR COMPOUNDS EIKONIZO THERAPEUTICS, INC. (US) 2022-03-24 US disclosed
US-20200171028-A1 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS HOLDINGS, LLC 2020-06-04 US disclosed
US-20200171028-A1 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS HOLDINGS, LLC 2020-06-04 US disclosed
US-10357493-B2 Metalloenzyme inhibitor compounds SELENITY THERAPEUTICS (BERMUDA), LTD. (BM) 2019-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240307391-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC1, HDAC2 CHRNA1 4120/4885CHRNG 3854/4885CHRNB1 4213/4885
US-20220088018-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC1, HDAC2 CHRNA1 4120/4885CHRNG 3854/4885CHRNB1 4213/4885
US-20200171028-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC1, HDAC2 CHRNA1 4120/4885CHRNG 3854/4885CHRNB1 4213/4885
US-20260124204-A1 METALLOENZYME INHIBITOR COMPOUNDS HDAC6, HDAC3, HDAC1 CHRNA1 428/4885CHRNG 378/4885CHRNB1 415/4885
US-11938134-B2 Metalloenzyme inhibitor compounds HDAC6, HDAC1, HDAC2 CHRNA1 4120/4885CHRNG 3854/4885CHRNB1 4213/4885
US-10357493-B2 Metalloenzyme inhibitor compounds HDAC6, HDAC1, HDAC2 CHRNA1 4120/4885CHRNG 3854/4885CHRNB1 4213/4885
US-12370194-B2 Metalloenzyme inhibitor compounds HDAC6, HDAC1, HDAC2 CHRNA1 4120/4885CHRNG 3854/4885CHRNB1 4213/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.