SCHEMBL21186166

SCHEMBL21186166

COc1ccnc(C(=O)Nc2nc3c(C)cc(Cl)cc3s2)c1O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
DCLK1 O15075 1/20 0.46
FES P07332 1/20 0.46
PIM1 P11309 1/20 0.46
CDK2 P24941 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
IRAK1 P51617 1/20 0.46
MAP4K2 Q12851 1/20 0.46
NTRK3 Q16288 1/20 0.46
HIPK4 Q8NE63 1/20 0.46
AURKB Q96GD4 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
STK17A Q9UEE5 1/20 0.46
MAP4K5 Q9Y4K4 1/20 0.46
CSNK1G3 Q9Y6M4 1/20 0.46
CHRM4 P08173 5/20 0.44
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21186172 0.90 NPC1 (0.55) NPC1RAB9ACHRM4KMT2AKDM4E
SCHEMBL21186164 0.89 RORC (0.46) NPC1RAB9ADCLK1FESPIM1
SCHEMBL21186013 0.84 RIPK1 (0.44) NPC1RAB9ACHRM4KMT2AKDM4E
SCHEMBL21186170 0.82 NPC1 (0.51) NPC1RAB9ACHRM4KMT2AKDM4E
SCHEMBL21186000 0.80 KMT2A (0.42) NPC1RAB9ACHRM4KMT2AKDM4E
SCHEMBL21186146 0.78 NPC1 (0.61) NPC1RAB9ADCLK1FESPIM1
SCHEMBL21186168 0.78 DCLK1 (0.53) NPC1RAB9ADCLK1FESPIM1
SCHEMBL21186121 0.78 NPC1 (0.43) NPC1RAB9ACHRM4KMT2AKDM4E
SCHEMBL21186175 0.77 DCLK1 (0.56) NPC1RAB9ADCLK1FESPIM1
SCHEMBL21186165 0.76 NPC1 (0.64) NPC1RAB9ADCLK1FESPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141980-A1 AGRICULTURAL CHEMICALS GLOBACHEM NV (BE) 2019-07-25 WO disclosed