SCHEMBL21187169

SCHEMBL21187169

CN(C)C1CNC(=O)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP3 Q9Y6F1 1/20 0.49
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
GPR3 P46089 1/20 0.41
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
SLC6A2 P23975 6/20 0.38
SLC6A4 P31645 6/20 0.38
PARP1 P09874 3/20 0.38
PDPK1 O15530 1/20 0.37
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
SLC6A3 Q01959 3/20 0.36
PBRM1 Q86U86 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12220005 0.77 PARP3 (0.53) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL6635520 0.77 PARP3 (0.53) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL21140586 0.74 SLC6A2 (0.39) GPR3SLC6A2SLC6A4SLC6A3
SCHEMBL11642624 0.73 CDK8 (0.51) PARP3HTR2AHTR2CHTR2B
SCHEMBL21187107 0.73 PARP3 (0.53) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL11750196 0.73 PARP3 (0.61) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL11130149 0.73 GPR3 (0.45) HTR2AHTR2CHTR2BGPR3SLC6A2
SCHEMBL21187216 0.72 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL8931375 0.72 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL29458586 0.72 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed