SCHEMBL21187134

SCHEMBL21187134

N=C(Nc1ccccc1F)NC1CCC(c2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
KMT2A Q03164 2/20 0.48
DGAT1 O75907 1/20 0.42
ALDH1A1 P00352 4/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
GRIN2B Q13224 1/20 0.40
EPHX2 P34913 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
LIPG Q9Y5X9 1/20 0.38
TRPV1 Q8NER1 2/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187111 0.80 NPC1 (0.45) NPC1RAB9AKMT2ADGAT1ALDH1A1
SCHEMBL21187139 0.80 NPC1 (0.45) NPC1RAB9AKMT2ADGAT1ALDH1A1
SCHEMBL21176799 0.75 KMT2A (0.43) NPC1RAB9AKMT2ADGAT1ALDH1A1
SCHEMBL21176800 0.75 KMT2A (0.43) NPC1RAB9AKMT2ADGAT1ALDH1A1
SCHEMBL21187113 0.75 IDO1 (0.55) NPC1RAB9AKMT2AALDH1A1L3MBTL1
SCHEMBL21187085 0.75 IDO1 (0.55) NPC1RAB9AKMT2AALDH1A1L3MBTL1
SCHEMBL16762704 0.74 LIPG (0.44) ALDH1A1L3MBTL1GRIN2BLIPG
SCHEMBL30050422 0.73 RAB9A (0.61) NPC1RAB9AKMT2AALDH1A1MEN1
SCHEMBL173455 0.73 RAB9A (0.61) NPC1RAB9AKMT2AALDH1A1MEN1
SCHEMBL21187119 0.72 NPC1 (0.51) NPC1RAB9AKMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed