SCHEMBL21187165

SCHEMBL21187165

COc1ccc(NC(=N)NC2CCC(c3cccc(F)c3)CC2)nc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 1/20 0.42
TRPV1 Q8NER1 9/20 0.40
HTR1A P08908 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
EP300 Q09472 1/20 0.37
CREBBP Q92793 1/20 0.37
ABL1 P00519 1/20 0.37
NTRK1 P04629 1/20 0.36
DPP4 P27487 1/20 0.36
IDO1 P14902 1/20 0.36
HDAC4 P56524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187095 0.87 KMT2A (0.41) KMT2APOLBMEN1TRPV1HTR1A
SCHEMBL21187129 0.72 RAB9A (0.49) POLB
SCHEMBL21187135 0.72 EPHX2 (0.40) KMT2APOLBMEN1TRPV1DPP4
SCHEMBL21187132 0.71 MAOA (0.48) KMT2A
SCHEMBL21187119 0.71 NPC1 (0.51) KMT2APOLBMEN1
SCHEMBL21187195 0.71 NPC1 (0.51) KMT2APOLBMEN1
SCHEMBL21187163 0.68 GRM5 (0.39) TRPV1DPP4
SCHEMBL1515236 0.66 HTR2C (0.47) HDAC4
SCHEMBL29878889 0.66 HTR2C (0.47) HDAC4
SCHEMBL21187149 0.65 NPC1 (0.46) KMT2APOLBMEN1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed