SCHEMBL21187358

SCHEMBL21187358

Cc1ncnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](N4C(=O)c5ccccc5C4O)CC3)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 6/20 0.35
MAPK1 P28482 3/20 0.35
TSHR P16473 3/20 0.35
CYP2C19 P33261 2/20 0.35
HIF1A Q16665 2/20 0.35
CLK4 Q9HAZ1 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
KMT2A Q03164 1/20 0.35
SYK P43405 1/20 0.34
POLB P06746 1/20 0.34
PRKDC P78527 1/20 0.34
ACVR1 Q04771 1/20 0.34
MAPT P10636 1/20 0.33
ERBB2 P04626 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28471532 0.86 ALDH1A1 (0.40) IRAK4L3MBTL1ALDH1A1MAPK1TSHR
SCHEMBL30817826 0.86 ALDH1A1 (0.40) IRAK4L3MBTL1ALDH1A1MAPK1TSHR
SCHEMBL21187359 0.86 ALDH1A1 (0.40) IRAK4L3MBTL1ALDH1A1MAPK1TSHR
SCHEMBL21187296 0.77 SYK (0.47) IRAK4HIF1ACLK4LMNACYP1A2
SCHEMBL30817825 0.77 SYK (0.47) IRAK4HIF1ACLK4LMNACYP1A2
SCHEMBL21178138 0.77 SYK (0.47) IRAK4HIF1ACLK4LMNACYP1A2
SCHEMBL21187340 0.75 IRAK4 (0.38) IRAK4HIF1ACLK4LMNACYP1A2
SCHEMBL21187331 0.72 MEN1 (0.38) IRAK4ALDH1A1MAPK1TSHRCYP2C19
SCHEMBL21178069 0.72 MEN1 (0.38) IRAK4ALDH1A1MAPK1TSHRCYP2C19
SCHEMBL30823285 0.72 MEN1 (0.38) IRAK4ALDH1A1MAPK1TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143678-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-07-25 WO disclosed