SCHEMBL21190850

SCHEMBL21190850

Fc1ccc(Oc2ccc(CBr)cc2Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 11/20 0.46
EPAS1 Q99814 2/20 0.39
PTGER4 P35408 1/20 0.39
PTGER2 P43116 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
HSPB1 P04792 1/20 0.38
PKM P14618 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21190859 0.87 TTR (0.50) NR3C1EPAS1PTGER4PTGER2PKM
SCHEMBL21191129 0.83 KDM4E (0.45) NR3C1SLC6A2SLC6A4SLC6A3
SCHEMBL21191013 0.83 TTR (0.53) NR3C1SLC6A2SLC6A4
SCHEMBL27689753 0.82 PKM (0.47) EPAS1SLC6A2SLC6A4SLC6A3HSPB1
SCHEMBL30444289 0.82 EPAS1 (0.52) NR3C1EPAS1HSPB1PKM
SCHEMBL15067971 0.82 EPAS1 (0.52) NR3C1EPAS1HSPB1PKM
SCHEMBL21190858 0.81 SLC6A4 (0.41) NR3C1EPAS1PTGER4PTGER2SLC6A2
SCHEMBL8695511 0.81 SLC6A4 (0.40) NR3C1PTGER4PTGER2SLC6A2SLC6A4
SCHEMBL21190854 0.79 BRD4 (0.50) NR3C1EPAS1SLC6A4
SCHEMBL12239036 0.79 ST14 (0.50) NR3C1SLC6A4PKMMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed