SCHEMBL21190854

SCHEMBL21190854

CS(=O)(=O)Cc1ccc(Oc2ccc(F)cc2)c(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.50
EPAS1 Q99814 7/20 0.45
SLC6A4 P31645 1/20 0.43
NR3C1 P04150 3/20 0.41
PTPN1 P18031 1/20 0.40
SOS1 Q07889 1/20 0.40
MET P08581 1/20 0.38
KDR P35968 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21191011 0.86 BRD4 (0.48) BRD4EPAS1NR3C1PTPN1CA2
SCHEMBL15067636 0.85 EPAS1 (0.55) BRD4EPAS1NR3C1METKDR
SCHEMBL30443821 0.85 EPAS1 (0.55) BRD4EPAS1NR3C1METKDR
SCHEMBL21681543 0.81 EPAS1 (0.41) BRD4EPAS1PTPN1KDR
SCHEMBL21190859 0.79 TTR (0.50) EPAS1NR3C1
SCHEMBL21190850 0.79 NR3C1 (0.46) EPAS1SLC6A4NR3C1
SCHEMBL30812017 0.77 THRA (0.46) BRD4EPAS1PTPN1
SCHEMBL27381068 0.77 THRA (0.46) BRD4EPAS1PTPN1
SCHEMBL21190858 0.77 SLC6A4 (0.41) EPAS1SLC6A4NR3C1
SCHEMBL21191065 0.76 BRD4 (0.54) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed