SCHEMBL21253552

SCHEMBL21253552

CC1Cn2c(nnc2-c2ccco2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 17/20 0.43
ABCB1 P08183 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20099682 1.00 P2RX7 (0.43) P2RX7ABCB1GPR119ADORA2AADORA1
SCHEMBL17596294 0.85 P2RX7 (0.50) P2RX7
SCHEMBL30980030 0.80 P2RX7 (0.56) P2RX7ABCB1GPR119ADORA2AADORA1
SCHEMBL17596276 0.79 P2RX7 (0.59) P2RX7
SCHEMBL17596277 0.79 P2RX7 (0.59) P2RX7
SCHEMBL17596464 0.77 P2RX7 (0.52) P2RX7GPR119
SCHEMBL17596463 0.77 P2RX7 (0.52) P2RX7GPR119
SCHEMBL17596300 0.76 P2RX7 (0.64) P2RX7GPR119
SCHEMBL17596299 0.76 P2RX7 (0.64) P2RX7GPR119
SCHEMBL17596616 0.75 P2RX7 (0.76) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191488-B1 P2X7 MODULATING N-ACYL-TRIAZOLOPYRAZINES JANSSEN PHARMACEUTICA NV (BE) 2019-08-14 EP disclosed