SCHEMBL21273015

SCHEMBL21273015

C=C(C)C(CC(=O)O)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21273013 1.00 SLC22A6 (0.33) SLC22A6TDP1SMN1; SMN2ALOX15MAPT
SCHEMBL14261039 0.80 SLC22A6 (0.35) SLC22A6TDP1SMN1; SMN2ALOX15MAPT
SCHEMBL11261532 0.78 SLC22A6 (0.30) SLC22A6
SCHEMBL11357843 0.78 ALDH1A1 (0.30) SLC22A6
SCHEMBL26444829 0.73 SLC22A6 (0.36) SLC22A6TDP1SMN1; SMN2
SCHEMBL21618444 0.72
SCHEMBL25242211 0.71 SLC22A6 (0.35) SLC22A6TDP1SMN1; SMN2
SCHEMBL11273231 0.71 ADRA1A (0.32)
SCHEMBL11268957 0.70 GABRR1 (0.38) SLC22A6TDP1SMN1; SMN2
SCHEMBL5184423 0.69 AAK1 (0.36) SLC22A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4026832-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 Almac Discovery Limited (GB) 2022-07-13 EP disclosed
US-10766903-B2 Piperidine derivatives as inhibitors of ubiquitin specific protease 7 ALMAC DISCOVERY LIMITED (GB) 2020-09-08 US disclosed
US-20190256518-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 GENETECH, INC. 2019-08-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190256518-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 USP7, USP5, UBA7 SLC22A6 4698/4885TDP1 1878/4885SMN1; SMN2 3429/4885
US-10766903-B2 Piperidine derivatives as inhibitors of ubiquitin specific protease 7 USP7, USP5, UBA7 SLC22A6 4698/4885TDP1 1878/4885SMN1; SMN2 3429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.