SCHEMBL21290152

SCHEMBL21290152

COc1cc(-c2cc(C)ccn2)ccc1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.57
KMO O15229 5/20 0.53
CCR1 P32246 1/20 0.48
CCR5 P51681 1/20 0.48
CCR8 P51685 1/20 0.48
KDM4C Q9H3R0 2/20 0.48
EGLN2 Q96KS0 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
USP2 O75604 1/20 0.45
POLB P06746 1/20 0.45
CYP2C9 P11712 1/20 0.45
ALOX12 P18054 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15345108 0.85 RAB9A (0.56) CCR1CCR5CCR8MEN1KMT2A
SCHEMBL16385281 0.81 RAB9A (0.57) KMOCCR1CCR5CCR8MEN1
SCHEMBL24257876 0.80 KMO (0.71) DYRK1AKMOEGLN2MEN1KMT2A
SCHEMBL21289970 0.79 DYRK1A (0.55) DYRK1AKMOKDM4CEGLN2MEN1
SCHEMBL21290163 0.78 KMO (0.50) DYRK1AKMOCCR1CCR5CCR8
SCHEMBL7241046 0.78 ALDH1A1 (0.56) CCR1CCR5CCR8MEN1KMT2A
SCHEMBL14758456 0.76 KMO (0.66) DYRK1AKMOKDM4CEGLN2MEN1
SCHEMBL27849397 0.76 DYRK1A (0.71) DYRK1AKMOKDM4CEGLN2ALDH1A1
SCHEMBL4302847 0.75 DYRK1A (0.65) DYRK1AKMOEGLN2MEN1KMT2A
SCHEMBL31695263 0.75 CCR1 (0.76) CCR1CCR5CCR8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed