SCHEMBL21290163

SCHEMBL21290163

COc1cc(-c2ccc(C)cn2)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.50
DYRK1A Q13627 1/20 0.50
CCR1 P32246 1/20 0.46
CCR5 P51681 1/20 0.46
CCR8 P51685 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
MAPT P10636 4/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
HPGD P15428 3/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 2/20 0.45
USP2 O75604 1/20 0.45
POLB P06746 1/20 0.45
CYP2C9 P11712 1/20 0.45
ALOX12 P18054 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KDM1A O60341 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14438065 0.85 RAB9A (0.56) CCR1CCR5CCR8HDAC6MAPT
SCHEMBL7604435 0.83 DYRK1A (0.56) KMODYRK1AMEN1KMT2AL3MBTL1
SCHEMBL16385283 0.81 MAPT (0.50) CCR1CCR5CCR8HDAC6MAPT
SCHEMBL6176031 0.80 IDO1 (0.46) KMODYRK1AKMT2AHPGDALDH1A1
SCHEMBL7684064 0.79 PSD (0.48) KMODYRK1AMAPTMEN1KMT2A
SCHEMBL12075586 0.78 RAB9A (0.57) CCR1CCR5CCR8HDAC6MAPT
SCHEMBL21290152 0.78 DYRK1A (0.57) KMODYRK1ACCR1CCR5CCR8
SCHEMBL27436349 0.78 ALDH1A1 (0.56) CCR1CCR5CCR8HDAC6MAPT
SCHEMBL30955276 0.78 ALDH1A1 (0.56) CCR1CCR5CCR8HDAC6MAPT
SCHEMBL23956247 0.77 KMO (0.47) KMODYRK1AMEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed