SCHEMBL21290159

SCHEMBL21290159

COc1cc(-c2ccc(Cl)cc2)ncc1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCL12 P48061 1/20 0.48
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
JAK2 O60674 1/20 0.43
EGFR P00533 1/20 0.43
CDK2 P24941 1/20 0.43
PIK3CA P42336 1/20 0.43
PIK3CB P42338 1/20 0.43
PIK3CG P48736 1/20 0.43
PTK2B Q14289 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
TDO2 P48775 5/20 0.41
IDO1 P14902 4/20 0.41
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290360 0.76 NPC1 (0.42) NPC1RAB9ATDO2IDO1MAPT
SCHEMBL458804 0.76 CYP3A4 (0.47) CYP1A2CYP3A4CYP2C19NPC1RAB9A
SCHEMBL16385279 0.74 KDM4E (0.48) CXCL12CYP1A2CYP3A4CYP2C19NPC1
SCHEMBL21290300 0.74 DGAT1 (0.46) NPC1RAB9ACASP3SENP7TDO2
SCHEMBL23956201 0.73 NPC1 (0.40) CYP3A4NPC1RAB9ATDO2IDO1
SCHEMBL23956221 0.73 TGFBR1 (0.42) CYP1A2CYP2C19NPC1RAB9ATDO2
SCHEMBL21586164 0.73 ERN1 (0.49) CXCL12CYP1A2CYP3A4CYP2C19ALOX5
SCHEMBL19780934 0.72 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C19NPC1RAB9A
SCHEMBL18015262 0.72 CYP1A2 (0.40) CYP1A2CYP3A4CYP2C19NPC1RAB9A
SCHEMBL1425419 0.72 S1PR1 (0.42) NPC1RAB9AMAPTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed