SCHEMBL21290168

SCHEMBL21290168

COc1cc(-c2cc(-c3ccccc3)c3ccccc3n2)ccc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 4/20 0.65
HPGD P15428 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 2/20 0.49
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 5/20 0.45
HTT P42858 2/20 0.45
MAPT P10636 2/20 0.45
L3MBTL1 Q9Y468 3/20 0.44
GAA P10253 1/20 0.44
DHODH Q02127 3/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPK1 P28482 2/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
ATM Q13315 1/20 0.43
HSD17B10 Q99714 1/20 0.43
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23956195 0.83 ACACA (0.43) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL23956229 0.83 KDM4E (0.62) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL23956151 0.81 L3MBTL1 (0.61) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL19050276 0.80 LIPG (0.59) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL12628400 0.80 LIPG (0.59) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL31707366 0.79 ACACA (1.00) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL16294371 0.79 ACACA (1.00) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL16203125 0.79 ACACA (0.49) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL21290172 0.78 L3MBTL1 (0.40) ACACAHPGDSMN1; SMN2LMNAALDH1A1
SCHEMBL21289786 0.76 ERN1 (0.43) HPGDSMN1; SMN2LMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed