SCHEMBL21290175

SCHEMBL21290175

COc1cccc(-c2ccc(B3OC(C)(C)C(C)(C)O3)cn2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.56
KDM1A O60341 1/20 0.48
SNCA P37840 1/20 0.45
LPL P06858 3/20 0.43
LIPG Q9Y5X9 3/20 0.43
DYRK1A Q13627 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
MAP4K4 O95819 1/20 0.40
FYN P06241 2/20 0.40
TDO2 P48775 1/20 0.39
CYP19A1 P11511 1/20 0.39
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21125910 0.88 DGAT1 (0.57) DGAT1LPLLIPG
SCHEMBL2697886 0.84 DGAT1 (0.67) DGAT1SNCALPLLIPGNPC1
SCHEMBL29688083 0.84 DGAT1 (0.67) DGAT1SNCALPLLIPGNPC1
SCHEMBL18015663 0.83 DGAT1 (0.59) DGAT1LPLLIPG
SCHEMBL21390894 0.83 DGAT1 (0.53) DGAT1KDM1ALPLLIPGCYP3A4
SCHEMBL15747744 0.82 DGAT1 (0.52) DGAT1LPLLIPGMAP4K4
SCHEMBL30739 0.81 DGAT1 (0.70) DGAT1LPLLIPG
SCHEMBL29688361 0.81 DGAT1 (0.70) DGAT1LPLLIPG
SCHEMBL15747886 0.80 DGAT1 (0.53) DGAT1LPLLIPGMAP4K4
SCHEMBL21290171 0.79 TOP1 (0.46) DGAT1KDM1ADYRK1ACLK4TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed