SCHEMBL21290171

SCHEMBL21290171

COc1cccc(-c2cc(-c3ccccc3)c(B3OC(C)(C)C(C)(C)O3)cn2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
DYRK1A Q13627 2/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
MAPK1 P28482 2/20 0.41
CYP2C19 P33261 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TP53 P04637 2/20 0.41
CLK4 Q9HAZ1 2/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
TGFBR1 P36897 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
KDM1A O60341 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18015456 0.86 LPL (0.46) NPC1RAB9ADYRK1AADORA2AADORA1
SCHEMBL20532210 0.81 LPL (0.42) NPC1RAB9ATSHRDGAT1SMN1; SMN2
SCHEMBL23956204 0.80 LIPG (0.41) NPC1RAB9AMAPK1HSD17B10TSHR
SCHEMBL21290175 0.79 DGAT1 (0.56) NPC1RAB9ADYRK1ACYP1A2CYP3A4
SCHEMBL21290177 0.79 IDO1 (0.45) NPC1RAB9AADORA1MAPK1HSD17B10
SCHEMBL25165559 0.77 LPL (0.45) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL18015448 0.74 LDHA (0.47) NPC1RAB9ACYP3A4DGAT1SMN1; SMN2
SCHEMBL21290348 0.74 TOP1 (0.53) TOP1NPC1RAB9ADYRK1AADORA2A
SCHEMBL12999308 0.73 LIPG (0.56) DGAT1TDO2
SCHEMBL19766305 0.72 LIPG (0.47) NPC1RAB9ADYRK1ADGAT1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed