SCHEMBL21292680

SCHEMBL21292680

O=C(NN=Cc1ccc(F)cc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 1.00
NPC1 O15118 6/20 1.00
SMN1; SMN2 Q16637 6/20 1.00
KMT2A Q03164 6/20 0.72
MEN1 O00255 5/20 0.72
POLB P06746 3/20 0.72
CYP1A2 P05177 2/20 0.72
CYP3A4 P08684 2/20 0.72
TDP1 Q9NUW8 2/20 0.72
CYP2D6 P10635 1/20 0.72
ESRRG P62508 2/20 0.70
ALDH1A1 P00352 1/20 0.68
MAPT P10636 1/20 0.68
PKM P14618 1/20 0.68
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA4 P22748 1/20 0.65
CA9 Q16790 1/20 0.65
CYP2C9 P11712 1/20 0.65
CYP2C19 P33261 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20115425 1.00 RAB9A (1.00) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL6720187 0.93 RAB9A (0.87) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL711754 0.90 RAB9A (0.81) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL711755 0.90 RAB9A (0.81) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL2830919 0.90 RAB9A (0.81) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL1563349 0.87 RAB9A (0.77) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL6634765 0.87 RAB9A (0.77) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL1563347 0.87 RAB9A (0.77) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL13568982 0.86 RAB9A (0.87) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL13475702 0.85 RAB9A (0.74) RAB9ANPC1SMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118307440-A Benzoyl hydrazone compound, synthesis method thereof, medicine containing compound and application of compound 泰州职业技术学院 2024-07-09 CN disclosed
CN-116396237-A Green synthesis method of oxadiazole compound 台州学院 2023-07-07 CN disclosed
CN-111848441-B N-substituted benzoyl hydrazone compound and preparation method and application thereof 山东中新科农生物科技有限公司 2023-02-17 CN disclosed
CN-111848441-A N-substituted benzoyl hydrazone compound and preparation method and application thereof 朱翠萍 2020-10-30 CN disclosed
US-10722489-B2 D-3-phosphoglycerate dehydrogenase allosteric inhibitor and use thereof PEKING UNIVERSITY (CN) 2020-07-28 US disclosed
US-20200054593-A1 D-3-PHOSPHOGLYCERATE DEHYDROGENASE ALLOSTERIC INHIBITOR AND USE THEREOF UNIV BEIJING (CN) 2020-02-20 US disclosed
US-20190262303-A1 D-3-PHOSPHOGLYCERATE DEHYDROGENASE ALLOSTERIC INHIBITOR AND USE THEREOF UNIV BEIJING (CN) 2019-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10722489-B2 D-3-phosphoglycerate dehydrogenase allosteric inhibitor and use thereof MDH2, MDH1, DLD RAB9A 4415/4885NPC1 4801/4885SMN1; SMN2 3566/4885
US-20200054593-A1 D-3-PHOSPHOGLYCERATE DEHYDROGENASE ALLOSTERIC INHIBITOR AND USE THEREOF MDH2, MDH1, DLD RAB9A 4415/4885NPC1 4801/4885SMN1; SMN2 3566/4885
US-20190262303-A1 D-3-PHOSPHOGLYCERATE DEHYDROGENASE ALLOSTERIC INHIBITOR AND USE THEREOF MDH2, MDH1, DLD RAB9A 4415/4885NPC1 4801/4885SMN1; SMN2 3566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.