SCHEMBL212959

SCHEMBL212959

O=CNc1nnc(-c2cccnc2)s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.60
NPC1 O15118 2/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
HDAC1 Q13547 2/20 0.51
HDAC2 Q92769 2/20 0.51
BLM P54132 2/20 0.49
HSD17B10 Q99714 5/20 0.48
MAPT P10636 2/20 0.47
TSHR P16473 2/20 0.47
CYP2A6 P11509 2/20 0.46
CYP2E1 P05181 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2B6 P20813 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP19A1 P11511 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13222434 0.82 CA1 (0.56) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL212851 0.80 KDM4E (0.61) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL1424931 0.79 KDM4E (0.75) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL174140 0.79 RAB9A (0.65) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL27768804 0.78 KDM4E (0.58) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL28148469 0.77 HPGDS (0.47) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL173422 0.75 KDM4E (0.67) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL174170 0.75 MEN1 (1.00) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL11008102 0.74 ALDH1A1 (0.53) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL9728291 0.74 CYP2A6 (0.42) RAB9ANPC1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed