SCHEMBL27768804

SCHEMBL27768804

O=Cc1nnc(-c2cccnc2)s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
CYP2A6 P11509 3/20 0.53
CYP3A4 P08684 3/20 0.53
CYP2E1 P05181 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2B6 P20813 2/20 0.53
CYP2C19 P33261 2/20 0.53
RAB9A P51151 3/20 0.51
NPC1 O15118 3/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
HSD17B10 Q99714 7/20 0.50
ALDH1A1 P00352 3/20 0.50
TSHR P16473 3/20 0.49
CYP19A1 P11511 1/20 0.46
AXL P30530 1/20 0.46
PBRM1 Q86U86 1/20 0.46
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1424931 0.82 KDM4E (0.75) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1
SCHEMBL27768554 0.79 KDM4E (0.53) KDM4ESMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL212959 0.78 RAB9A (0.60) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1
SCHEMBL12278703 0.75 KDM4E (0.66) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1
SCHEMBL255577 0.75 KDM4E (0.66) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1
SCHEMBL30803985 0.75 KDM4E (0.66) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1
SCHEMBL1680233 0.75 HSD17B10 (0.55) KDM4ESMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL27790186 0.75 CYP2A6 (0.58) CYP2A6CYP3A4CYP2E1CYP2C9CYP2B6
SCHEMBL27817490 0.74 KDM4E (0.51) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1
SCHEMBL970073 0.74 KDM4E (0.64) KDM4ESMN1; SMN2CYP2A6CYP3A4CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed